Structure-based mechanism of cysteinyl leukotriene receptor inhibition by antiasthmatic drugs A Luginina*, A Gusach*, E Marin, A Mishin, R Brouillette, P Popov, ... Science advances 5 (10), eaax2518, 2019 | 76 | 2019 |
Structural basis of ligand selectivity and disease mutations in cysteinyl leukotriene receptors A Gusach*, A Luginina*, E Marin, RL Brouillette, É Besserer-Offroy, ... Nature communications 10 (1), 1-9, 2019 | 62 | 2019 |
Beyond structure: emerging approaches to study GPCR dynamics A Gusach, I Maslov, A Luginina, V Borshchevskiy, A Mishin, V Cherezov Current Opinion in Structural Biology 63, 18-25, 2020 | 50 | 2020 |
An outlook on using serial femtosecond crystallography in drug discovery A Mishin, A Gusach, A Luginina, E Marin, V Borshchevskiy, V Cherezov Expert Opinion on Drug Discovery 14 (9), 933-945, 2019 | 29 | 2019 |
Metabolic fate of human immunoactive sterols in Mycobacterium tuberculosis T Varaksa, S Bukhdruker, I Grabovec, E Marin, A Kavaleuski, A Gusach, ... Journal of molecular biology 433 (4), 166763, 2021 | 23 | 2021 |
Structure-based virtual screening of ultra-large library yields potent antagonists for a lipid GPCR AA Sadybekov, RL Brouillette, E Marin, AV Sadybekov, A Luginina, ... Biomolecules 10 (12), 1634, 2020 | 23 | 2020 |
Sub-millisecond conformational dynamics of the A2A adenosine receptor revealed by single-molecule FRET I Maslov, O Volkov, P Khorn, P Orekhov, A Gusach, P Kuzmichev, ... Communications Biology 6 (1), 362, 2023 | 18 | 2023 |
Hydroxylation of antitubercular drug candidate, SQ109, by mycobacterial cytochrome P450 S Bukhdruker, T Varaksa, I Grabovec, E Marin, P Shabunya, M Kadukova, ... International journal of molecular sciences 21 (20), 7683, 2020 | 15 | 2020 |
New insights into GPCR coupling and dimerisation from cryo-EM structures A Gusach, J García-Nafría, CG Tate Current Opinion in Structural Biology 80, 102574, 2023 | 10 | 2023 |
Structural basis for receptor selectivity and inverse agonism in S1P5 receptors E Lyapina*, E Marin*, A Gusach*, P Orekhov, A Gerasimov, A Luginina, ... Nature communications 13 (1), 1-14, 2022 | 10 | 2022 |
Small-wedge synchrotron and serial XFEL datasets for Cysteinyl leukotriene GPCRs E Marin, A Luginina, A Gusach, K Kovalev, S Bukhdruker, P Khorn, ... Scientific data 7 (1), 388, 2020 | 5 | 2020 |
Molecular recognition of an aversive odorant by the murine trace amine-associated receptor TAAR7f A Gusach, Y Lee, AN Khoshgrudi, E Mukhaleva, N Ma, EJ Koers, Q Chen, ... bioRxiv, 2023 | 1 | 2023 |
Successful GPCR structure determination using PAL XFEL E Marin, A Gusach, A Luginina, K Kovalev, W Liu, U Weierstall, HK Nam, ... JOURNAL OF BIOENERGETICS AND BIOMEMBRANES 50 (6), 513-513, 2018 | 1 | 2018 |
Structural diversity of leukotriene G-protein coupled receptors A Luginina, A Gusach, E Lyapina, P Khorn, N Safronova, M Shevtsov, ... Journal of Biological Chemistry, 105247, 2023 | | 2023 |