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Georgi Stavrakov
Georgi Stavrakov
Faculty of Pharmacy, Medical University of Sofia
Verified email at orgchm.bas.bg
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Cited by
Year
Galantamine derivatives with indole moiety: Docking, design, synthesis and acetylcholinesterase inhibitory activity
M Atanasova, G Stavrakov, I Philipova, D Zheleva, N Yordanov, ...
Bioorganic & Medicinal Chemistry 23 (17), 5382-5389, 2015
822015
Theophylline-7-acetic acid derivatives with amino acids as anti-tuberculosis agents
Y Voynikov, V Valcheva, G Momekov, P Peikov, G Stavrakov
Bioorganic & medicinal chemistry letters 24 (14), 3043-3045, 2014
532014
Novel camphane-based anti-tuberculosis agents with nanomolar activity
G Stavrakov, V Valcheva, I Philipova, I Doytchinova
European Journal of Medicinal Chemistry 70, 372-379, 2013
442013
Novel hits for acetylcholinesterase inhibition derived by docking-based screening on ZINC database
I Doytchinova, M Atanasova, I Valkova, G Stavrakov, I Philipova, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 33 (1), 768-776, 2018
372018
Docking‐based design and synthesis of galantamine–camphane hybrids as inhibitors of acetylcholinesterase
G Stavrakov, I Philipova, D Zheleva‐Dimitrova, I Valkova, E Salamanova, ...
Chemical Biology & Drug Design 90 (5), 709-718, 2017
332017
Synthetic piperine amide analogs with antimycobacterial activity
I Philipova, V Valcheva, R Mihaylova, M Mateeva, I Doytchinova, ...
Chemical Biology & Drug Design 91 (3), 763-768, 2018
322018
Synthesis and antimycobacterial activity of novel camphane-based agents
G Stavrakov, I Philipova, V Valcheva, G Momekov
Bioorganic & Medicinal Chemistry Letters 24 (1), 165-167, 2014
302014
Synthesis of ferrocene-based amido-phosphine ligands via highly diastereoselective ortho-lithiation and their application in Pd-catalyzed asymmetric allylic …
I Philipova, G Stavrakov, A Chimov, R Nikolova, B Shivachev, V Dimitrov
Tetrahedron: Asymmetry 22 (9), 970-979, 2011
282011
Antimycobacterial activity of chiral aminoalcohols with camphane scaffold
Z Petkova, V Valcheva, G Momekov, P Petrov, V Dimitrov, I Doytchinova, ...
European Journal of Medicinal Chemistry 81, 150-157, 2014
252014
A novel galantamine-curcumin hybrid as a potential multi-target agent against neurodegenerative disorders
R Simeonova, D Zheleva, I Valkova, G Stavrakov, I Philipova, ...
Molecules 26 (7), 1865, 2021
232021
Galantamine-curcumin hybrids as dual-site binding acetylcholinesterase inhibitors
G Stavrakov, I Philipova, A Lukarski, M Atanasova, D Zheleva, ...
Molecules 25 (15), 3341, 2020
232020
Docking‐based Design of Galantamine Derivatives with Dual‐site Binding to Acetylcholinesterase
G Stavrakov, I Philipova, D Zheleva, M Atanasova, S Konstantinov, ...
Molecular informatics 35 (6-7), 278-285, 2016
232016
From Central to Axial to Central Chirality: Enantioselective Construction of the trans‐4,5,9,10‐Tetrahydroxy‐9,10‐dihydrophenanthrene System
G Stavrakov, M Keller, B Breit
European Journal of Organic Chemistry 2007 (34), 5726-5733, 2007
232007
Cytisine as a scaffold for ortho-diphenylphosphinobenzenecarboxamide ligands for Pd-catalyzed asymmetric allylic alkylation
I Philipova, G Stavrakov, N Vassilev, R Nikolova, B Shivachev, V Dimitrov
Journal of Organometallic Chemistry 778, 10-20, 2015
212015
Design, Synthesis, and Antimycobacterial Activity of Novel Theophylline‐7‐Acetic Acid Derivatives With Amino Acid Moieties
G Stavrakov, V Valcheva, Y Voynikov, I Philipova, M Atanasova, ...
Chemical Biology & Drug Design 87 (3), 335-341, 2016
192016
Highly diastereoselective ortho-lithiation of chiral ferrocenecarboxamides
G Stavrakov, I Philipova, B Ivanova, V Dimitrov
Tetrahedron: Asymmetry 21 (15), 1845-1854, 2010
192010
Synthesis and absolute configuration of planar chiral ferrocenophanes by amide-directed ortho-lithiation
G Stavrakov, S Simova, V Dimitrov
Tetrahedron: Asymmetry 19 (18), 2119-2122, 2008
152008
Camphane-based phosphino-carboxamide ligands as P, O-chelates in Pd-catalyzed enantioselective allylic alkylation
I Philipova, G Stavrakov, V Dimitrov
Tetrahedron: Asymmetry 23 (13), 927-930, 2012
132012
Pyrazinamide-Pharmaceutical, biochemical and pharmacological properties and reappraisal of its role in the chemotherapy of tuberculosis
G Momekov, D Ferdinandov, Y Voynikov, G Stavrakov, P Peykov
Pharmacia 61 (1), 38-67, 2014
122014
Cytotoxicity assay on several theophylline-7-acetic acid amides with amino acids
Y Voynikov, G Momekov, P Peikov, G Stavrakov
Pharmacia 61, 12-16, 2014
112014
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