Galantamine derivatives with indole moiety: Docking, design, synthesis and acetylcholinesterase inhibitory activity M Atanasova, G Stavrakov, I Philipova, D Zheleva, N Yordanov, ... Bioorganic & Medicinal Chemistry 23 (17), 5382-5389, 2015 | 82 | 2015 |
Theophylline-7-acetic acid derivatives with amino acids as anti-tuberculosis agents Y Voynikov, V Valcheva, G Momekov, P Peikov, G Stavrakov Bioorganic & medicinal chemistry letters 24 (14), 3043-3045, 2014 | 53 | 2014 |
Novel camphane-based anti-tuberculosis agents with nanomolar activity G Stavrakov, V Valcheva, I Philipova, I Doytchinova European Journal of Medicinal Chemistry 70, 372-379, 2013 | 44 | 2013 |
Novel hits for acetylcholinesterase inhibition derived by docking-based screening on ZINC database I Doytchinova, M Atanasova, I Valkova, G Stavrakov, I Philipova, ... Journal of Enzyme Inhibition and Medicinal Chemistry 33 (1), 768-776, 2018 | 37 | 2018 |
Docking‐based design and synthesis of galantamine–camphane hybrids as inhibitors of acetylcholinesterase G Stavrakov, I Philipova, D Zheleva‐Dimitrova, I Valkova, E Salamanova, ... Chemical Biology & Drug Design 90 (5), 709-718, 2017 | 33 | 2017 |
Synthetic piperine amide analogs with antimycobacterial activity I Philipova, V Valcheva, R Mihaylova, M Mateeva, I Doytchinova, ... Chemical Biology & Drug Design 91 (3), 763-768, 2018 | 32 | 2018 |
Synthesis and antimycobacterial activity of novel camphane-based agents G Stavrakov, I Philipova, V Valcheva, G Momekov Bioorganic & Medicinal Chemistry Letters 24 (1), 165-167, 2014 | 30 | 2014 |
Synthesis of ferrocene-based amido-phosphine ligands via highly diastereoselective ortho-lithiation and their application in Pd-catalyzed asymmetric allylic … I Philipova, G Stavrakov, A Chimov, R Nikolova, B Shivachev, V Dimitrov Tetrahedron: Asymmetry 22 (9), 970-979, 2011 | 28 | 2011 |
Antimycobacterial activity of chiral aminoalcohols with camphane scaffold Z Petkova, V Valcheva, G Momekov, P Petrov, V Dimitrov, I Doytchinova, ... European Journal of Medicinal Chemistry 81, 150-157, 2014 | 25 | 2014 |
A novel galantamine-curcumin hybrid as a potential multi-target agent against neurodegenerative disorders R Simeonova, D Zheleva, I Valkova, G Stavrakov, I Philipova, ... Molecules 26 (7), 1865, 2021 | 23 | 2021 |
Galantamine-curcumin hybrids as dual-site binding acetylcholinesterase inhibitors G Stavrakov, I Philipova, A Lukarski, M Atanasova, D Zheleva, ... Molecules 25 (15), 3341, 2020 | 23 | 2020 |
Docking‐based Design of Galantamine Derivatives with Dual‐site Binding to Acetylcholinesterase G Stavrakov, I Philipova, D Zheleva, M Atanasova, S Konstantinov, ... Molecular informatics 35 (6-7), 278-285, 2016 | 23 | 2016 |
From Central to Axial to Central Chirality: Enantioselective Construction of the trans‐4,5,9,10‐Tetrahydroxy‐9,10‐dihydrophenanthrene System G Stavrakov, M Keller, B Breit European Journal of Organic Chemistry 2007 (34), 5726-5733, 2007 | 23 | 2007 |
Cytisine as a scaffold for ortho-diphenylphosphinobenzenecarboxamide ligands for Pd-catalyzed asymmetric allylic alkylation I Philipova, G Stavrakov, N Vassilev, R Nikolova, B Shivachev, V Dimitrov Journal of Organometallic Chemistry 778, 10-20, 2015 | 21 | 2015 |
Design, Synthesis, and Antimycobacterial Activity of Novel Theophylline‐7‐Acetic Acid Derivatives With Amino Acid Moieties G Stavrakov, V Valcheva, Y Voynikov, I Philipova, M Atanasova, ... Chemical Biology & Drug Design 87 (3), 335-341, 2016 | 19 | 2016 |
Highly diastereoselective ortho-lithiation of chiral ferrocenecarboxamides G Stavrakov, I Philipova, B Ivanova, V Dimitrov Tetrahedron: Asymmetry 21 (15), 1845-1854, 2010 | 19 | 2010 |
Synthesis and absolute configuration of planar chiral ferrocenophanes by amide-directed ortho-lithiation G Stavrakov, S Simova, V Dimitrov Tetrahedron: Asymmetry 19 (18), 2119-2122, 2008 | 15 | 2008 |
Camphane-based phosphino-carboxamide ligands as P, O-chelates in Pd-catalyzed enantioselective allylic alkylation I Philipova, G Stavrakov, V Dimitrov Tetrahedron: Asymmetry 23 (13), 927-930, 2012 | 13 | 2012 |
Pyrazinamide-Pharmaceutical, biochemical and pharmacological properties and reappraisal of its role in the chemotherapy of tuberculosis G Momekov, D Ferdinandov, Y Voynikov, G Stavrakov, P Peykov Pharmacia 61 (1), 38-67, 2014 | 12 | 2014 |
Cytotoxicity assay on several theophylline-7-acetic acid amides with amino acids Y Voynikov, G Momekov, P Peikov, G Stavrakov Pharmacia 61, 12-16, 2014 | 11 | 2014 |